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CYCLIC COMPOUND HAVING SELECTIVE KRAS INHIBITORY EFFECT ON HRAS AND NRAS

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CYCLIC COMPOUND HAVING SELECTIVE KRAS INHIBITORY EFFECT ON HRAS AND NRAS

PCT NATIONAL PHASE APPLICATION

Published

date

Filed on 6 November 2024

Abstract

The present inventors found a cyclic compound that selectively inhibits KRAS. The present inventors also found that the cyclic compound interacts with a KRAS-specific amino acid residue.

Patent Information

Application ID202447084925
Invention FieldCHEMICAL
Date of Application06/11/2024
Publication Number47/2024

Inventors

NameAddressCountryNationality
KAWADA Hatsuoc/o CHUGAI SEIYAKU KABUSHIKI KAISHA, 200, Kajiwara, Kamakura-shi, Kanagawa 2478530JapanJapan
TAKANO Kojic/o CHUGAI SEIYAKU KABUSHIKI KAISHA, 200, Kajiwara, Kamakura-shi, Kanagawa 2478530JapanJapan
KOTAKE Tomoyac/o CHUGAI SEIYAKU KABUSHIKI KAISHA, 135, Komakado 1-chome, Gotemba-shi, Shizuoka 4128513JapanJapan
KAGE Miraic/o CHUGAI SEIYAKU KABUSHIKI KAISHA, 135, Komakado 1-chome, Gotemba-shi, Shizuoka 4128513JapanJapan
HASHIMOTO Satoshic/o CHUGAI SEIYAKU KABUSHIKI KAISHA, 135, Komakado 1-chome, Gotemba-shi, Shizuoka 4128513JapanJapan
TAMIYA Minoruc/o CHUGAI SEIYAKU KABUSHIKI KAISHA, 200, Kajiwara, Kamakura-shi, Kanagawa 2478530JapanJapan
WAKAMIYA Yumac/o CHUGAI SEIYAKU KABUSHIKI KAISHA, 200, Kajiwara, Kamakura-shi, Kanagawa 2478530JapanJapan
HAYASHI Ryujic/o CHUGAI SEIYAKU KABUSHIKI KAISHA, 200, Kajiwara, Kamakura-shi, Kanagawa 2478530JapanJapan
MORITA Yuyac/o CHUGAI SEIYAKU KABUSHIKI KAISHA, 200, Kajiwara, Kamakura-shi, Kanagawa 2478530JapanJapan

Applicants

NameAddressCountryNationality
CHUGAI SEIYAKU KABUSHIKI KAISHA5-1, Ukima 5-chome, Kita-ku, Tokyo 1158543JapanJapan

Documents

NameDate
202447084925-FORM-26 [07-11-2024(online)].pdf07/11/2024
202447084925-COMPLETE SPECIFICATION [06-11-2024(online)].pdf06/11/2024
202447084925-DECLARATION OF INVENTORSHIP (FORM 5) [06-11-2024(online)].pdf06/11/2024
202447084925-FORM 1 [06-11-2024(online)].pdf06/11/2024
202447084925-FORM 18 [06-11-2024(online)].pdf06/11/2024
202447084925-NOTIFICATION OF INT. APPLN. NO. & FILING DATE (PCT-RO-105-PCT Pamphlet) [06-11-2024(online)].pdf06/11/2024
202447084925-PRIORITY DOCUMENTS [06-11-2024(online)].pdf06/11/2024
202447084925-PROOF OF RIGHT [06-11-2024(online)].pdf06/11/2024
202447084925-REQUEST FOR EXAMINATION (FORM-18) [06-11-2024(online)].pdf06/11/2024
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